{"id":12551,"date":"2022-03-31T09:39:16","date_gmt":"2022-03-31T07:39:16","guid":{"rendered":"https:\/\/dignitynews.eu\/?p=12551"},"modified":"2022-03-31T09:39:16","modified_gmt":"2022-03-31T07:39:16","slug":"w-gdansku-poszukuja-zwiazkow-ktore-pomoga-opracowac-nowy-lek-na-covid-19","status":"publish","type":"post","link":"https:\/\/dignitynews.eu\/pl\/w-gdansku-poszukuja-zwiazkow-ktore-pomoga-opracowac-nowy-lek-na-covid-19\/","title":{"rendered":"W Gda\u0144sku poszukuj\u0105 zwi\u0105zk\u00f3w, kt\u00f3re pomog\u0105 opracowa\u0107 nowy lek na COVID-19"},"content":{"rendered":"<h5>Naukowcy z Politechniki Gda\u0144skiej (PG) pracuj\u0105 nad otrzymaniem nowych zwi\u0105zk\u00f3w blokuj\u0105cych dzia\u0142anie enzym\u00f3w odgrywaj\u0105cych kluczow\u0105 rol\u0119 w procesie namna\u017cania koronawirusa SARS-CoV-2. W niedalekiej przysz\u0142o\u015bci ma to pozwoli\u0107 na opracowanie skutecznego, bezpiecznego i taniego polskiego leku eliminuj\u0105cego ci\u0119\u017cki przebieg COVID-19 &#8211; informuje uczelnia.<\/h5>\n<p>Celem bada\u0144 jest otrzymanie nowych, skutecznych inhibitor\u00f3w enzymu proteazy SARS-CoV-2 Mpro, czyli niskocz\u0105steczkowych zwi\u0105zk\u00f3w chemicznych blokuj\u0105cych jej dzia\u0142anie. Enzym ten jest wytwarzany w ludzkich kom\u00f3rkach zainfekowanych koronawirusem i odgrywa kluczow\u0105 rol\u0119 w procesie replikacji koronawirusa SARS-CoV-2, odpowiedzialnego za pandemi\u0119 COVID-19.<\/p>\n<p>Naukowcy z gda\u0144skiej uczelni licz\u0105, \u017ce otrzymanie nowych inhibitor\u00f3w enzymu pozwoli w niedalekiej przysz\u0142o\u015bci na opracowanie skutecznego, taniego, polskiego leku, eliminuj\u0105cego ci\u0119\u017cki przebieg choroby, kt\u00f3ry b\u0119dzie mo\u017cna stosowa\u0107 doustnie. Wst\u0119pne badania s\u0105 obiecuj\u0105ce, a odkryte dotychczas zwi\u0105zki mog\u0105 nie wykazywa\u0107 niepo\u017c\u0105danych dzia\u0142a\u0144 ubocznych.<\/p>\n<p>W pierwszym etapie badacze, wykorzystuj\u0105c komputerowe techniki modelowania molekularnego, zaprojektowali struktury zwi\u0105zk\u00f3w o najwy\u017cszym stopniu dopasowania do miejsca aktywnego proteazy.<\/p>\n<p>&#8211; Substancje chemiczne klasyfikowane jako inhibitory proteazy s\u0105 zaliczane do jednych z najnowocze\u015bniejszych i niezwykle obiecuj\u0105cych strategii projektowania nowych lek\u00f3w stosowanych w wielu terapiach przeciwwirusowych, w tym w leczeniu COVID-19, i s\u0105 skutecznym uzupe\u0142nieniem szczepie\u0144 oraz innych dzia\u0142a\u0144 profilaktycznych &#8211; t\u0142umaczy kierownik zespo\u0142u badawczego, dr hab. in\u017c. Sebastian Demkowicz, prof. PG z Katedry Chemii Organicznej.<\/p>\n<p>Arkadiusz S\u0142omczy\u0144ski<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Naukowcy z Politechniki Gda\u0144skiej (PG) pracuj\u0105 nad otrzymaniem nowych zwi\u0105zk\u00f3w blokuj\u0105cych dzia\u0142anie enzym\u00f3w odgrywaj\u0105cych kluczow\u0105 rol\u0119 w procesie namna\u017cania koronawirusa SARS-CoV-2. W niedalekiej przysz\u0142o\u015bci ma to pozwoli\u0107 na opracowanie skutecznego,&hellip;<\/p>\n","protected":false},"author":7,"featured_media":12552,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_mi_skip_tracking":false,"footnotes":""},"categories":[49],"tags":[],"class_list":["post-12551","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-nauka"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v19.4 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>W Gda\u0144sku poszukuj\u0105 zwi\u0105zk\u00f3w, kt\u00f3re pomog\u0105 opracowa\u0107 nowy lek na COVID-19 - Godno\u015b\u0107 - DignityNews.eu<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/dignitynews.eu\/pl\/w-gdansku-poszukuja-zwiazkow-ktore-pomoga-opracowac-nowy-lek-na-covid-19\/\" \/>\n<meta property=\"og:locale\" content=\"pl_PL\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"W Gda\u0144sku poszukuj\u0105 zwi\u0105zk\u00f3w, kt\u00f3re pomog\u0105 opracowa\u0107 nowy lek na COVID-19 - Godno\u015b\u0107 - DignityNews.eu\" \/>\n<meta property=\"og:description\" content=\"Naukowcy z Politechniki Gda\u0144skiej (PG) pracuj\u0105 nad otrzymaniem nowych zwi\u0105zk\u00f3w blokuj\u0105cych dzia\u0142anie enzym\u00f3w odgrywaj\u0105cych kluczow\u0105 rol\u0119 w procesie namna\u017cania koronawirusa SARS-CoV-2. 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